SCHEMBL5828246

SCHEMBL5828246

COc1ccc2[nH]c(C(C)=Cc3ccccc3)cc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
HDAC6 Q9UBN7 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2C9 P11712 1/20 0.60
TSHR P16473 1/20 0.60
FLT3 P36888 6/20 0.58
PDGFRB P09619 2/20 0.58
PDGFRA P16234 2/20 0.58
KDM4E B2RXH2 4/20 0.53
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
MAPT P10636 2/20 0.52
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828241 1.00 MEN1 (0.60) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829080 0.84 MEN1 (0.64) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829074 0.84 MEN1 (0.64) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829078 0.84 MEN1 (0.64) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5827564 0.83 MEN1 (0.56) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5827563 0.83 MEN1 (0.56) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829672 0.77 MEN1 (0.69) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829674 0.77 MEN1 (0.69) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL5829677 0.77 MEN1 (0.69) MEN1KMT2AHDAC6CYP1A2CYP3A4
SCHEMBL2729934 0.75 PDGFRB (0.79) MEN1KMT2AHDAC6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed