SCHEMBL5840409

SCHEMBL5840409

CCn1cnc2c(Nc3cc(C(F)(F)F)cc(C(F)(F)F)c3)nc(N[C@H]3CC[C@H](O)CC3)nc21

nearest known ligand 0.83

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 17/20 0.83
PRKCA P17252 4/20 0.56
SRC P12931 1/20 0.52
CCNB2 O95067 1/20 0.52
CCNB1 P14635 1/20 0.52
CCNB3 Q8WWL7 1/20 0.52
PDGFRA P16234 2/20 0.51
CCNE1 P24864 2/20 0.51
CDK2 P24941 2/20 0.51
EGFR P00533 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5840414 1.00 CDK1 (0.83) CDK1PRKCASRCCCNB2CCNB1
SCHEMBL5839065 0.91 CDK1 (1.00) CDK1PRKCACCNB2CCNB1CCNB3
SCHEMBL5839069 0.91 CDK1 (1.00) CDK1PRKCACCNB2CCNB1CCNB3
SCHEMBL5839489 0.91 CDK1 (0.83) CDK1PRKCAPDGFRACCNE1CDK2
SCHEMBL5840941 0.91 CDK1 (0.82) CDK1PRKCASRCPDGFRACCNE1
SCHEMBL5840934 0.91 CDK1 (0.82) CDK1PRKCASRCPDGFRACCNE1
SCHEMBL5840461 0.91 CDK1 (0.83) CDK1PRKCAPDGFRACCNE1CDK2
SCHEMBL5839495 0.91 CDK1 (0.83) CDK1PRKCAPDGFRACCNE1CDK2
SCHEMBL5840330 0.85 CDK1 (1.00) CDK1PRKCASRCPDGFRACCNE1
SCHEMBL5840337 0.85 CDK1 (1.00) CDK1PRKCASRCPDGFRACCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed