SCHEMBL5847751

SCHEMBL5847751

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(F)c(F)c3)cc3c1N2CCC3

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MMP13 P45452 1/20 0.39
HTR2A P28223 5/20 0.39
HTR2C P28335 5/20 0.39
HTR2B P41595 1/20 0.39
GPR119 Q8TDV5 6/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
USP30 Q70CQ3 2/20 0.38
DRD2 P14416 2/20 0.37
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
SLC6A4 P31645 1/20 0.37
DPP4 P27487 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847077 0.97 NPC1 (0.40) NPC1RAB9AMMP13HTR2AHTR2C
SCHEMBL5847308 0.89 USP30 (0.41) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL5846966 0.89 HTR2A (0.43) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL5846974 0.88 NPC1 (0.40) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL5847223 0.88 HTR2C (0.41) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL5846980 0.87 STS (0.41) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL5846954 0.87 TP53 (0.42) NPC1RAB9AUSP30
SCHEMBL5848083 0.87 USP30 (0.40) NPC1RAB9AGPR119PTPN2PTPN1
SCHEMBL5847354 0.86 HTR2A (0.44) NPC1RAB9AHTR2AHTR2CGPR119
SCHEMBL5415767 0.86 HTR2C (0.41) HTR2AHTR2CHTR2BDRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed