SCHEMBL5854355

SCHEMBL5854355

CSc1ccccc1C(=O)C1CCN(c2ccnc3ccc(-c4cn(C(c5ccccc5)(c5ccccc5)c5ccccc5)nc4C(F)(F)F)cc23)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
ITGB2 P05107 4/20 0.35
ICAM1 P05362 4/20 0.35
ITGAL P20701 4/20 0.35
MELK Q14680 2/20 0.35
SLC22A12 Q96S37 2/20 0.34
CYP8B1 Q9UNU6 5/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
MTOR P42345 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5851864 0.88 CYP3A4 (0.38) CYP3A4HPGDITGB2ICAM1ITGAL
SCHEMBL3848141 0.87 CYP3A4 (0.50) CYP3A4HPGDITGB2ICAM1ITGAL
SCHEMBL3845276 0.83 CYP3A4 (0.37) CYP3A4HPGDCYP8B1LMNAKMT2A
SCHEMBL3848728 0.81 CHRM4 (0.39) CYP3A4HPGDCYP8B1MTORKMT2A
SCHEMBL3852739 0.81 CHRM4 (0.43) CYP3A4HPGDCYP8B1
SCHEMBL3845503 0.80 CYP3A4 (0.40) CYP3A4HPGDLMNAPKMMTOR
SCHEMBL3855550 0.80 CYP3A4 (0.37) CYP3A4HPGDITGB2ICAM1ITGAL
SCHEMBL3846231 0.80 MAPKAPK2 (0.46) CYP3A4HPGDLMNAKMT2A
SCHEMBL3850111 0.79 MTOR (0.39) MTORKMT2A
SCHEMBL3846799 0.79 MTOR (0.40) CYP3A4HPGDSLC22A12CYP8B1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed