SCHEMBL5854786

SCHEMBL5854786

CCCC(NC(=O)C(F)(F)F)N(Cc1ccc2c(c1)NC(=O)C(C)O2)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.42
SMYD3 Q9H7B4 4/20 0.36
KDR P35968 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5470810 0.95 PARP1 (0.41) PARP1SMYD3KDRHSD17B10PDE3B
SCHEMBL5472751 0.91 PARP1 (0.33) PARP1
SCHEMBL5464744 0.87 PARP1 (0.47) PARP1SMYD3KDRHSD17B10
SCHEMBL5474592 0.86 PARP1 (0.45) PARP1SMYD3KDRHSD17B10
SCHEMBL5467227 0.84 PARP1 (0.32) PARP1HSD17B10
SCHEMBL5465466 0.82 PARP1 (0.44) PARP1SMYD3KDRHSD17B10
SCHEMBL5482158 0.82 KDM4E (0.30)
SCHEMBL5471766 0.79 PARP1 (0.51) PARP1SMYD3KDRHSD17B10PDE3B
SCHEMBL5472790 0.78 PARP1 (0.36) PARP1HSD17B10
SCHEMBL7711130 0.78 PARP1 (0.53) PARP1SMYD3HSD17B10PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141566-B1 Benzoxazine and benzothiazine derivatives and the use thereof in medicaments SCHERING AKTIENGESELLSCHAFT (DE) 2006-11-28 US disclosed