SCHEMBL5855043

SCHEMBL5855043

CC1(c2ccc(O)cc2)COc2cc(O)ccc2C1COCCCCCCC[S+]([O-])CCCC(F)(F)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.34
TMEM97 Q5BJF2 2/20 0.32
HTR2B P41595 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
NR1I2 O75469 1/20 0.30
NR3C1 P04150 1/20 0.30
PGR P06401 1/20 0.30
ESRRA P11474 1/20 0.30
EPHX2 P34913 1/20 0.30
PPARG P37231 1/20 0.30
ESR2 Q92731 1/20 0.30
NR1H4 Q96RI1 1/20 0.30
SIRT5 Q9NXA8 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5854261 0.94 ESR1 (0.34) ESR1TMEM97HTR2BSIGMAR1NR1I2
SCHEMBL5854386 0.92 ESR1 (0.33) ESR1TMEM97HTR2BSIGMAR1NR1I2
SCHEMBL7588501 0.89 ESR1 (0.34) ESR1TMEM97HTR2BSIGMAR1NR1I2
SCHEMBL7589349 0.89 ESR1 (0.34) ESR1TMEM97HTR2BSIGMAR1NR1I2
SCHEMBL5854250 0.85 TMEM97 (0.30) ESR1TMEM97NR1I2NR3C1PGR
SCHEMBL5854257 0.84 ESR1 (0.31) ESR1
SCHEMBL5855127 0.84 ESR1 (0.34) ESR1NR1I2NR3C1PGRESRRA
SCHEMBL5856278 0.84 ESR1 (0.33) ESR1TMEM97HTR2BSIGMAR1NR1I2
SCHEMBL7589074 0.84 ESR1 (0.36) ESR1ESR2CYP3A4ALOX15
SCHEMBL5854246 0.83 ESR1 (0.33) ESR1TMEM97NR1I2NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074819-B2 Benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2006-07-11 US disclosed
US-6645951-B1 Antiestrogens for treating breast cancer CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-11-11 US disclosed