SCHEMBL5856958

SCHEMBL5856958

COc1ccc2c(c1)OCC(C)(c1cccnc1)C2CCCCCCCCCSCCCC(F)(F)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.34
HTR1A P08908 1/20 0.31
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
CTSD P07339 1/20 0.31
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5855951 0.90 CYP19A1 (0.33) HTR1AHTR2BSIGMAR1CYP19A1
SCHEMBL5857506 0.83 BACE1 (0.38) BACE1HTR1AHTR2BSIGMAR1CTSD
SCHEMBL7588543 0.83 PTPN1 (0.31)
SCHEMBL7587357 0.83 PTPN1 (0.31)
SCHEMBL5855979 0.82 ESR1 (0.38) HTR1AHTR2BSIGMAR1
SCHEMBL5854301 0.81 BACE1 (0.35) BACE1HTR1AHTR2BSIGMAR1CTSD
SCHEMBL5854227 0.80 ESR1 (0.33) HTR2BSIGMAR1
SCHEMBL5857401 0.79 HTR2B (0.33) HTR1AHTR2BSIGMAR1
SCHEMBL7585889 0.78 ESR1 (0.36) HTR2BSIGMAR1
SCHEMBL7588656 0.78 ESR1 (0.36) HTR2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074819-B2 Benzopyran or thiobenzopyran derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2006-07-11 US disclosed
US-6645951-B1 Antiestrogens for treating breast cancer CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-11-11 US disclosed
EP-1087959-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-04-04 EP disclosed
WO-1999065893-A1 NOVEL BENZOPYRAN OR THIOBENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1999-12-23 WO disclosed