SCHEMBL5861548

SCHEMBL5861548

CC(C)N1CCN(c2ccc(Nc3nc(N)c(C(=O)c4ccc(OCC(F)F)cc4)s3)cc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 10/20 0.68
CCND1 P24385 10/20 0.68
CCNT1 O60563 8/20 0.58
CDK9 P50750 8/20 0.58
CDK6 Q00534 8/20 0.58
CDK11A Q9UQ88 7/20 0.58
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
NPC1 O15118 2/20 0.55
CDK5 Q00535 3/20 0.50
CDK5R1 Q15078 2/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
GSK3A P49840 2/20 0.49
GSK3B P49841 2/20 0.49
LTK P29376 1/20 0.49
CLK2 P49760 1/20 0.49
CDK7 P50613 1/20 0.49
LIMK1 P53667 1/20 0.49
PRKCQ Q04759 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5741662 0.90 CDK4 (0.72) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5742997 0.85 CDK4 (0.72) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5741691 0.84 CDK4 (0.71) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5743010 0.84 CDK4 (0.70) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5742969 0.83 CDK4 (0.71) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5743054 0.83 CDK4 (0.85) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5743411 0.83 CDK4 (0.87) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5744236 0.82 CDK4 (0.66) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5743586 0.82 CDK4 (0.75) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL5743774 0.82 CDK4 (0.72) CDK4CCND1CCNT1CDK9CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094896-B2 Diaminothiazoles having antiproliferative activity HOFFMANN-LA ROCHE INC. (US) 2006-08-22 US disclosed