SCHEMBL5869486

SCHEMBL5869486

O=C(O)C(Cc1ccccc1)NC(Cc1cncn1Cc1ccccc1)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACE2 Q9BYF1 4/20 0.62
ACE P12821 3/20 0.62
CYP11B1 P15538 7/20 0.54
CYP11B2 P19099 7/20 0.54
MME P08473 1/20 0.47
IDO1 P14902 1/20 0.47
FNTA P49354 2/20 0.45
FNTB P49356 2/20 0.45
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
TSHR P16473 1/20 0.44
TRHDE Q9UKU6 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
AGTR2 P50052 1/20 0.42
HPGDS O60760 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8250261 1.00 ACE2 (0.62) ACE2ACECYP11B1CYP11B2MME
SCHEMBL7222649 0.91 ACE2 (0.62) ACE2ACECYP11B1CYP11B2IDO1
SCHEMBL8248307 0.91 ACE2 (0.62) ACE2ACECYP11B1CYP11B2IDO1
SCHEMBL5870208 0.89 ACE2 (0.78) ACE2ACECYP11B1CYP11B2MME
SCHEMBL8248569 0.89 ACE2 (0.78) ACE2ACECYP11B1CYP11B2MME
SCHEMBL8249070 0.87 ACE (0.58) ACE2ACECYP11B1CYP11B2MME
SCHEMBL5869812 0.87 ACE (0.58) ACE2ACECYP11B1CYP11B2MME
SCHEMBL5870473 0.84 ACE2 (0.57) ACE2ACECYP11B1CYP11B2MME
SCHEMBL8249532 0.84 ACE (0.70) ACE2ACECYP11B1CYP11B2MME
SCHEMBL5869403 0.84 ACE (0.70) ACE2ACECYP11B1CYP11B2MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6632830-B1 Blood pressure related disease or disorder, cell proliferation disorder, kidney disorder, kinetensin associated disorder, inflammation associated disorder, or an allergic disorder MILLENNIUM PHARMACEUTICALS, INC. 2003-10-14 US claimed
US-7045532-B2 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-05-16 US disclosed
US-6632830-B1 Blood pressure related disease or disorder, cell proliferation disorder, kidney disorder, kinetensin associated disorder, inflammation associated disorder, or an allergic disorder MILLENNIUM PHARMACEUTICALS, INC. 2003-10-14 US disclosed