SCHEMBL5887399

SCHEMBL5887399

CCOc1ccc(-n2nc(CC(C(=O)O)c3cccc(Cl)c3)cc2-c2ccc3c(c2)OCO3)cc1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 16/20 0.65
SLC16A3 O15427 1/20 0.49
SLC16A1 P53985 1/20 0.49
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
BCL2 P10415 2/20 0.42
MDM2 Q00987 2/20 0.42
MCL1 Q07820 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4015199 0.87 CCKAR (0.71) CCKARPTGS2BCL2MDM2MCL1
SCHEMBL4005841 0.86 CCKAR (0.70) CCKARBCL2MDM2MCL1
SCHEMBL4009018 0.85 CCKAR (0.74) CCKARSLC16A3SLC16A1PTGS1PTGS2
SCHEMBL13980038 0.80 CCKAR (0.64) CCKARSLC16A3SLC16A1PTGS1PTGS2
SCHEMBL4137399 0.79 CCKAR (1.00) CCKARPTGS2
SCHEMBL4014758 0.79 CCKAR (0.60) CCKARSLC16A3SLC16A1PTGS1PTGS2
SCHEMBL4858502 0.78 CCKAR (1.00) CCKARPTGS1PTGS2
SCHEMBL4005418 0.78 CCKAR (0.74) CCKARSLC16A3SLC16A1PTGS2
SCHEMBL4012786 0.78 CCKAR (0.60) CCKARPTGS1PTGS2
SCHEMBL4007905 0.78 CCKAR (0.60) CCKARPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US disclosed