SCHEMBL5889188

SCHEMBL5889188

COc1c(Nc2ncc(C#N)s2)ncnc1N1CCN(CC(=O)NC(C)C)CC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.47
CYP11B2 P19099 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889233 0.89 KDR (0.47) KDRCYP11B2KDM4EALDH1A1SMN1; SMN2
SCHEMBL5889027 0.89 KDR (0.47) KDRCYP11B2KDM4EALDH1A1SMN1; SMN2
SCHEMBL5889112 0.81 KDR (0.69) KDR
SCHEMBL5889031 0.76 KDR (0.44) KDR
SCHEMBL5889026 0.76 KDR (0.44) KDR
SCHEMBL5889124 0.76 KDR (0.69) KDRCYP11B2KDM4EALDH1A1SMN1; SMN2
SCHEMBL5889024 0.75 KDR (0.54) KDRAURKA
SCHEMBL5889195 0.70 KDR (0.72) KDR
SCHEMBL5889115 0.69 KDR (0.65) KDRAURKA
SCHEMBL5889238 0.69 KDR (0.68) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115597-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2006-10-03 US disclosed