SCHEMBL5889254

SCHEMBL5889254

N#Cc1cnc(Nc2cc(N3CCC(C(=O)O)CC3)ncn2)s1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.74
CHEK1 O14757 1/20 0.45
KIT P10721 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889186 0.85 KDR (1.00) KDRCHEK1
SCHEMBL5889166 0.83 KDR (0.83) KDRCHEK1KIT
SCHEMBL5889049 0.82 KDR (0.73) KDRKIT
SCHEMBL5889168 0.82 KDR (0.81) KDRCHEK1KIT
SCHEMBL5889069 0.82 KDR (1.00) KDRKIT
SCHEMBL5889039 0.81 KDR (1.00) KDRCHEK1KIT
SCHEMBL6800930 0.81 KDR (1.00) KDRCHEK1
SCHEMBL5889162 0.81 KDR (0.67) KDRKIT
SCHEMBL7691786 0.81 KDR (0.76) KDRKIT
SCHEMBL6802538 0.81 KDR (0.76) KDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115597-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2006-10-03 US disclosed