SCHEMBL5896641

SCHEMBL5896641

N=C(N)CCNC(=O)c1cc(NC(=O)c2ccc(C(=O)NCCN)cc2)cn1CC1CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRAS P01112 13/20 0.48
ESR1 P03372 13/20 0.48
ESR2 Q92731 13/20 0.48
TOP1 P11387 2/20 0.48
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
HIF1A Q16665 1/20 0.47
ITGB3 P05106 3/20 0.39
ITGA2B P08514 3/20 0.39
CYP1A2 P05177 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
MAOB P27338 1/20 0.37
TERT O14746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889504 0.95 HRAS (0.52) HRASESR1ESR2TOP1KDM4E
SCHEMBL5896854 0.92 HRAS (0.48) HRASESR1ESR2TOP1KDM4E
SCHEMBL5889463 0.86 HRAS (0.46) HRASESR1ESR2TOP1KDM4E
SCHEMBL5680577 0.86 HRAS (0.44) HRASESR1ESR2TOP1KDM4E
SCHEMBL5889617 0.85 HRAS (0.50) HRASESR1ESR2TOP1KDM4E
SCHEMBL7177291 0.85 HRAS (0.39) HRASESR1ESR2TOP1KDM4E
SCHEMBL5896846 0.84 TOP1 (0.45) HRASESR1ESR2TOP1KDM4E
SCHEMBL5889611 0.82 HRAS (0.49) HRASESR1ESR2TOP1KDM4E
SCHEMBL5889829 0.80 HRAS (0.48) HRASESR1ESR2TOP1KDM4E
SCHEMBL5889570 0.76 MAP3K5 (0.38) HRASESR1ESR2TOP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141680-B2 Aromatic compounds possessing antifungal or antibacterial activity GENELABS TECHNOLOGIES, INC. 2006-11-28 US disclosed