Dutasteride

Dutasteride

SCHEMBL5903

C[C@]12C=CC(=O)N[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](C(=O)Nc3cc(C(F)(F)F)ccc3C(F)(F)F)CC[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SRD5A1SRD5A2SRD5A3

The experimentally established mechanism targets of Dutasteride. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A1 known ✓ P18405 19/20 1.00
SRD5A2 known ✓ P31213 8/20 1.00
LMNA P02545 1/20 1.00
ABCB11 O95342 1/20 1.00
GLRA1 P23415 1/20 1.00
KEAP1 Q14145 1/20 1.00
NFE2L2 Q16236 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dutasteride SCHEMBL1832772 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL1285958 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL9975973 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL1108295 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL13495828 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL997007 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL10028296 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL12194984 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL20776136 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1
Dutasteride SCHEMBL4775587 1.00 SRD5A1 (1.00) SRD5A1SRD5A2LMNAABCB11GLRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 13005 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107401-A2 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY OF POLYLACTIC ACID FOR HAIR GROWTH DURAIRAJ KALPNA KAY (US) 2026-05-21 WO claimed
US-20260115207-A1 COUMARIN-MODIFIED ANDROGENS FOR THE TREATMENT OF PROSTATE CANCER HEALTH RESEARCH INC (US) 2026-04-30 US claimed
US-12599613-B2 Composition comprising dutasteride CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2026-04-14 US claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
US-12582651-B2 Pharmaceutical composition comprising tadalafil or pharmaceutically acceptable salt thereof and dutasteride or pharmaceutically acceptable salt thereof exhibiting novel dissolution rate DONG KOOK PHARM. CO., LTD. (KR) 2026-03-24 US claimed
US-12582601-B2 Orodispersible powder composition BIOPHARMA SYNERGIES, S.L. (ES) 2026-03-24 US claimed
US-20260076981-A1 HAIR REGROWTH TOPICAL COMPOSITION SPEIER GARY J (US) 2026-03-19 US claimed
US-20260060913-A1 BIOACTIVE WALNUT PEPTIDES FOR TREATING HAIR LOSS L'OREAL (FR) 2026-03-05 US claimed
US-20260060936-A1 INDOLIUM-BASED STABILIZERS OF HYDROPHOBIC DRUGS TECHNION RES & DEV FOUNDATION (IL) 2026-03-05 US claimed
EP-4698175-A1 LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR, COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-02-25 EP claimed
EP-1173141-A1 SHAMPOOS PROVIDING A SUPERIOR COMBINATION OF ANTI-DANDRUFF EFFICACY AND CONDITIONING The Procter & Gamble Company (US) 2002-01-23 EP claimed
US-20010048942-A1 Dutasteride to prevent and treat atherosclerosis WEISMAN KENNETH (US) 2001-12-06 US claimed
US-20010047022-A1 Treatment or prevention of prostate cancer with a COX-2 selective inhibiting drug MERCK & CO., INC. 2001-11-29 US claimed
US-20010041713-A1 Treatment or prevention of prostate cancer with a COX-2 selective inhibiting drug WALDSTREICHER JOANNE (US) 2001-11-15 US claimed
WO-2001060365-A1 TREATMENT OR PREVENTION OF PROSTATE CANCER WITH A COX-2 SELECTIVE INHIBITING DRUG MERCK & CO., INC. (US) 2001-08-23 WO claimed
WO-2001054688-A1 TREATMENT OR PREVENTION OF PROSTATE CANCER WITH A COX-2 SELECTIVE INHIBITING DRUG MERCK & CO., INC. (US) 2001-08-02 WO claimed
WO-2000066072-A1 SHAMPOOS PROVIDING A SUPERIOR COMBINATION OF ANTI-DANDRUFF EFFICACY AND CONDITIONING THE PROCTER & GAMBLE COMPANY (US) 2000-11-09 WO claimed
WO-1999036030-A2 PHARMACEUTICAL COMPOSITION AND METHOD FOR TREATING DI-HYDROXYTESTOSTERONE DEPENDENT CONDITIONS DAVITZ, MICHAEL, A. (US) 1999-07-22 WO claimed
EP-0859617-A1 METHOD OF PREVENTING ANDROGENETIC ALOPECIA WITH 5-ALPHA REDUCTASE INHIBITORS Merck & Co., Inc. (US) 1998-08-26 EP claimed
WO-1997011702-A1 METHOD OF PREVENTING ANDROGENETIC ALOPECIA WITH 5-ALPHA REDUCTASE INHIBITORS MERCK & CO., INC. (US) 1997-04-03 WO claimed