SCHEMBL5956864

SCHEMBL5956864

C#Cc1ccc(NC(=O)N2CCC[C@@H]2C(=O)Nc2ccc(N3CCOCC3=O)c(C)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 2/20 0.49
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.47
F10 P00742 4/20 0.46
NPSR1 Q6W5P4 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76669 0.89 F10 (0.57) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL76587 0.89 F10 (0.57) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL76586 0.89 F10 (0.57) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL5956859 0.88 F10 (0.57) MEN1KMT2ACYP2C9CYP2C19TSHR
SCHEMBL5956956 0.88 F10 (0.61) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL76844 0.86 F10 (0.56) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL76845 0.86 F10 (0.56) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL5956913 0.86 F10 (0.54) MEN1KMT2ATSHRF10
SCHEMBL4450787 0.85 F10 (0.50) F10
SCHEMBL5956960 0.84 F10 (0.65) MEN1KMT2AF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633346-B1 PYRROLIDIN-1, 2- DICARBOXYLIC ACID- 1- (4- ETHINYL- PHENYL) - AMID|- 2- (PHENYL)- AMID| DERIVATIVE AS INHIBITORS OF COAGULATION FACTOR XA AND VIIA FOR THE TREATMENT OF THROMBOSIS MERCK PATENT GMBH (DE) 2006-08-23 EP claimed