SCHEMBL5966467

SCHEMBL5966467

Cc1cc(Br)ccc1C(=O)NS(=O)(=O)c1cnc(C(C)C)s1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 7/20 0.52
FLT4 P35916 7/20 0.52
KDR P35968 7/20 0.52
GPR27 Q9NS67 1/20 0.40
FBP1 P09467 7/20 0.39
EGFR P00533 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
NLRP3 Q96P20 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5966436 0.86 FLT1 (0.56) FLT1FLT4KDRGPR27FBP1
SCHEMBL5966435 0.79 FLT1 (0.53) FLT1FLT4KDR
SCHEMBL5966459 0.77 FLT1 (0.60) FLT1FLT4KDRGPR27NLRP3
SCHEMBL5966688 0.76 FLT1 (0.58) FLT1FLT4KDRGPR27EGFR
SCHEMBL5966458 0.76 FLT1 (0.61) FLT1FLT4KDRGPR27EGFR
SCHEMBL31310538 0.75 FLT1 (0.56) FLT1FLT4KDREGFRNLRP3
SCHEMBL5186222 0.74 FLT1 (0.50) FLT1FLT4KDRGPR27FBP1
SCHEMBL5966503 0.73 FLT1 (0.54) FLT1FLT4KDRGPR27FBP1
SCHEMBL5966440 0.73 FLT1 (0.54) FLT1FLT4KDRGPR27EGFR
SCHEMBL5966617 0.73 FLT1 (0.57) FLT1FLT4KDRGPR27EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1298709-C Thiophene-amd thiazolesulfonamides as antineoplastic agents LILLY CO ELI (US) 2007-02-07 CN disclosed
EP-1442030-B1 THIOPENE- AMD THIAZOLESULFONAMIDES AS ANTINEOPLASTIC AGENTS LILLY CO ELI (US) 2006-08-30 EP disclosed
CN-1575286-A Thiophene-amd thiazolesulfonamides as antineoplastic agents LILLY CO ELI (US) 2005-02-02 CN disclosed