SCHEMBL5969742

SCHEMBL5969742

CCN(CC)C(=O)Oc1ccc(C[C@H](NC(=O)[C@@H]2CCC(=O)N2Cc2ccc(C#N)cc2)C(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.58
ITGA4 P13612 10/20 0.58
CAPN1 P07384 4/20 0.45
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5681725 0.92 ITGB1 (0.53) ITGB1ITGA4CAPN1KMT2AKDM4E
SCHEMBL5679669 0.82 ITGB1 (0.63) ITGB1ITGA4CAPN1ALDH1A1
SCHEMBL5163741 0.82 CAPN1 (0.44) ITGB1ITGA4CAPN1KMT2A
SCHEMBL5693902 0.81 ITGB1 (0.55) ITGB1ITGA4CAPN1KMT2AKDM4E
SCHEMBL5679763 0.81 ITGB1 (0.55) ITGB1ITGA4CAPN1KMT2AALDH1A1
SCHEMBL5166690 0.79 ITGB1 (0.47) ITGB1ITGA4CAPN1ITGB3ITGA2B
SCHEMBL5693874 0.78 ITGB1 (0.52) ITGB1ITGA4CAPN1KMT2A
SCHEMBL5164182 0.76 ITGB1 (0.74) ITGB1ITGA4CAPN1
SCHEMBL5165158 0.76 ITGB1 (0.74) ITGB1ITGA4CAPN1
SCHEMBL5165080 0.76 CAPN1 (0.56) ITGB1ITGA4CAPN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7101855-B2 Pyroglutamic acid derivatives and related compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-09-05 US claimed