SCHEMBL598206

SCHEMBL598206

COC(C)NCC(=O)O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047031 0.81 EGLN1 (0.35)
SCHEMBL4063978 0.80 EGLN1 (0.34)
SCHEMBL161143 0.79
SCHEMBL16267760 0.77
SCHEMBL31198195 0.77
Hydrochloric Acid SCHEMBL5595965 0.77
SCHEMBL16267390 0.77
SCHEMBL19883542 0.76
SCHEMBL7432682 0.74 CA14 (0.45)
SCHEMBL7429510 0.74 CA14 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 85 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748439-A2 A PEPTOID-PEPTIDE HYBRID, NMEG-ALPHA-CGRP, AND ITS USE IN CARDIOVASCULAR DISEASES University of South Carolina (US) 2026-05-27 EP claimed
US-12533421-B2 Methods for making multilayered vesicles THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2026-01-27 US claimed
CN-115361961-A Method for preventing or treating pancreatic dysfunction or diabetes by up-regulating human cathepsin LL-37 to inhibit islet amyloid polypeptide (IAPP) self-assembly 斯坦福大学托管董事会 2022-11-18 CN claimed
US-20220257791-A1 METHODS FOR MAKING MULTILAYERED VESICLES THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND 2022-08-18 US claimed
US-20220257711-A1 PEPTOID-PEPTIDE HYBRID, NMEG-aCGRP, AND ITS USE IN CARDIOVASCULAR DISEASES UNIVERSITY OF SOUTH CAROLINA (US) 2022-08-18 US claimed
EP-3996733-A1 A PEPTOID-PEPTIDE HYBRID, NMEG-ACGRP, AND ITS USE IN CARDIOVASCULAR DISEASES University of South Carolina (US) 2022-05-18 EP claimed
WO-2021022117-A1 A PEPTOID-PEPTIDE HYBRID, NMEG-ACGRP, AND ITS USE IN CARDIOVASCULAR DISEASES UNIVERSITY OF SOUTH CAROLINA (US) 2021-02-04 WO claimed
US-10676509-B2 Surface-immobilized antimicrobial peptoids NORTHWESTERN UNIVERSITY (US) 2020-06-09 US claimed
US-20180051056-A1 SYNTHETIC MINIATURE PROTEIN SCAFFOLDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME KIRSHENBAUM KENT (US) 2018-02-22 US claimed
US-8114599-B2 Using multiplexed single-base extension assays comprising monodisperse uncharged polyamides conjugated to preferential nucleotide sequences for genotyping samples NORTHWESTERN UNIVERSITY (US) 2012-02-14 US claimed
JP-2010527270-A 2010-08-12 JP claimed
EP-2155276-A2 MEDICAL DEVICES HAVING ANTIFOULING CHARACTER Boston Scientific Scimed, Inc. (US) 2010-02-24 EP claimed
US-20090286435-A1 Method for Producing, and a Substrate with, a Surface with Specific Characteristics SURFACE INNOVATIONS LIMITED (GB) 2009-11-19 US claimed
WO-2008144392-A2 MEDICAL DEVICES HAVING ANTIFOULING CHARACTER BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-11-27 WO claimed
US-7371533-B2 Methods for separation of polymeric compounds UNIVERSITY OF OTTAWA (CA) 2008-05-13 US claimed
EP-1868739-A2 METHOD FOR PRODUCING, AND A SUBSTRATE WITH, A SURFACE WITH SPECIFIC CHARACTERISTICS UNIVERSITY OF DURHAM (GB) 2007-12-26 EP claimed
US-20070215472-A1 Electroosmotic flow for end labelled free solution electrophoresis UNIVERSITY OF OTTAWA (CA) 2007-09-20 US claimed
WO-2006109055-A2 METHOD FOR COATING A SUBSTRATE TO GIVE PROTEIN RESISTANCE AND COATED SUBSTRATE UNIVERSITY OF DURHAM (GB) 2006-10-19 WO claimed
US-20060177840-A1 Methods for separation of polymeric compounds DOE-DEITR 2006-08-10 US claimed
EP-4748439-A2 A PEPTOID-PEPTIDE HYBRID, NMEG-ALPHA-CGRP, AND ITS USE IN CARDIOVASCULAR DISEASES University of South Carolina (US) 2026-05-27 EP disclosed
US-12533421-B2 Methods for making multilayered vesicles THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2026-01-27 US disclosed
EP-3183365-B1 REUSABLE INITIATORS FOR SYNTHESIZING NUCLEIC ACIDS MOLECULAR ASSEMBLIES INC (US) 2025-10-15 EP disclosed
US-12397057-B2 Hydrophobically modified polypeptoids and uses thereof THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2025-08-26 US disclosed
WO-2025043073-A1 METHODS AND MATERIALS FOR SYNTHESIZING POLYNUCLEOTIDES Molecular Assemblies, Inc. (US) 2025-02-27 WO disclosed
US-12168211-B2 Reusable initiators for synthesizing nucleic acids Molecular Assemblies, Inc. (US) 2024-12-17 US disclosed
US-12152265-B2 Reusable initiators for synthesizing nucleic acids Molecular Assemblies, Inc. (US) 2024-11-26 US disclosed
US-20240268768-A1 Method of Preventing or Treating Pancreatic Dysfunction or Diabetes by Upregulating Human Cathelicidin LL-37 to Inhibit Islet Amyloid Polypeptide (IAPP) Self-Assembly THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-08-15 US disclosed
US-20240165245-A1 MULTIVALENT PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME NEW YORK UNIVERSITY (US) 2024-05-23 US disclosed
CN-117693353-A Cell-permeable cyclic peptides and uses thereof 安奈彻产品股份有限公司 2024-03-12 CN disclosed
US-20230302145-A1 SURFACTANT PROTEIN C MIMICS DISPLAYING PATHOGEN- OR ALLERGEN-BINDING MOIETIES Maxwell Biosciences, Inc. 2023-09-28 US disclosed
US-11766480-B2 Multivalent peptoid oligomers, pharmaceutical compositions and methods of using same NEW YORK UNIVERSITY (US) 2023-09-26 US disclosed
US-20230227880-A1 REUSABLE INITIATORS FOR SYNTHESIZING NUCLEIC ACIDS Molecular Assemblies, Inc. 2023-07-20 US disclosed
CN-116406280-A Surfactant protein C mimetics exhibiting pathogen or allergen binding moieties 安纳利斯·E·巴隆 2023-07-07 CN disclosed
CN-116096882-A Reusable initiator for synthesizing nucleic acid 分子组装公司 2023-05-09 CN disclosed
US-20230103381-A1 REUSABLE INITIATORS FOR SYNTHESIZING NUCLEIC ACIDS Molecular Assemblies, Inc. 2023-04-06 US disclosed
EP-4149509-A1 SURFACTANT PROTEIN C MIMICS DISPLAYING PATHOGEN- OR ALLERGEN-BINDING MOIETIES Barron, Annelise E. (US) 2023-03-22 EP disclosed
EP-4133070-A1 REUSABLE INITIATORS FOR SYNTHESIZING NUCLEIC ACIDS Molecular Assemblies, Inc. (US) 2023-02-15 EP disclosed
CN-115361961-A Method for preventing or treating pancreatic dysfunction or diabetes by up-regulating human cathepsin LL-37 to inhibit islet amyloid polypeptide (IAPP) self-assembly 斯坦福大学托管董事会 2022-11-18 CN disclosed
CN-115297883-A Cell permeable cyclic peptides and uses thereof 安奈彻产品股份有限公司 2022-11-04 CN disclosed
US-20220257711-A1 PEPTOID-PEPTIDE HYBRID, NMEG-aCGRP, AND ITS USE IN CARDIOVASCULAR DISEASES UNIVERSITY OF SOUTH CAROLINA (US) 2022-08-18 US disclosed
US-20220257791-A1 METHODS FOR MAKING MULTILAYERED VESICLES THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND 2022-08-18 US disclosed
US-11384377-B2 Reusable initiators for synthesizing nucleic acids Molecular Assemblies, Inc. (US) 2022-07-12 US disclosed
EP-3996733-A1 A PEPTOID-PEPTIDE HYBRID, NMEG-ACGRP, AND ITS USE IN CARDIOVASCULAR DISEASES University of South Carolina (US) 2022-05-18 EP disclosed
US-11331643-B2 Reusable initiators for synthesizing nucleic acids Molecular Assemblies, Inc. (US) 2022-05-17 US disclosed
US-20220072135-A1 HYDROPHOBICALLY MODIFIED POLYPEPTOIDS AND USES THEREOF THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND 2022-03-10 US disclosed
WO-2021231343-A1 SURFACTANT PROTEIN C MIMICS DISPLAYING PATHOGEN- OR ALLERGEN-BINDING MOIETIES BARRON ANNELISE E (US) 2021-11-18 WO disclosed
US-20210040539-A1 METHODS AND SYSTEMS FOR DETECTING TARGET NUCLEIC ACIDS BASHKIROV VLADIMIR I (US) 2021-02-11 US disclosed
WO-2021022117-A1 A PEPTOID-PEPTIDE HYBRID, NMEG-ACGRP, AND ITS USE IN CARDIOVASCULAR DISEASES UNIVERSITY OF SOUTH CAROLINA (US) 2021-02-04 WO disclosed
US-10676509-B2 Surface-immobilized antimicrobial peptoids NORTHWESTERN UNIVERSITY (US) 2020-06-09 US disclosed
US-10421954-B2 Hybrid polymers, pharmaceutical compositions and methods of synthesizing the same NEW YORK UNIVERSITY (US) 2019-09-24 US disclosed
EP-3417059-A1 METHODS AND SYSTEMS FOR DETECTING TARGET NUCLEIC ACIDS Bashkirov, Vladimir I. (US) 2018-12-26 EP disclosed
CN-109072225-A METHODS AND SYSTEMS FOR DETECTING TARGET NUCLEIC ACIDS 弗拉迪米尔.I.巴什基洛夫 2018-12-21 CN disclosed
US-20180311367-A1 MULTIVALENT PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME UNIV NEW YORK (US) 2018-11-01 US disclosed
EP-3356397-A1 TREATMENT OF BONE GROWTH DISORDERS Fondazione Telethon (IT) 2018-08-08 EP disclosed
US-20180051056-A1 SYNTHETIC MINIATURE PROTEIN SCAFFOLDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME KIRSHENBAUM KENT (US) 2018-02-22 US disclosed
US-20180030519-A1 METHODS AND SYSTEMS FOR DETECTING TARGET NUCLEIC ACIDS BASHKIROV VLADIMIR I (US) 2018-02-01 US disclosed
WO-2017143317-A1 METHODS AND SYSTEMS FOR DETECTING TARGET NUCLEIC ACIDS BASHKIROV VLADIMIR I (US) 2017-08-24 WO disclosed
US-20170015991-A1 HYBRID POLYMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF SYNTHESIZING THE SAME NEW YORK UNIVERSITY 2017-01-19 US disclosed
US-20160376646-A1 NUCLEIC ACID SEQUENCING IN FREE SOLUTION USING PROTEIN POLYMER DRAG-TAGS NORTHWESTERN UNIVERSITY 2016-12-29 US disclosed
US-9458449-B2 Hybrid polymers, pharmaceutical compositions and methods of synthesizing the same NEW YORK UNIVERSITY (US) 2016-10-04 US disclosed
EP-2976353-A1 AUTOPHAGY-INDUCING PEPTIDE ANALOGS The Board of Regents, University of Texas System (US) 2016-01-27 EP disclosed
US-20150126450-A1 MULTIVALENT PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME NEW YORK UNIVERSITY 2015-05-07 US disclosed
US-20150044189-A1 HYBRID POLYMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF SYNTHESIZING THE SAME NEW YORK UNIVERSITY 2015-02-12 US disclosed
EP-1814976-B1 PEPTIDOMIMETIC POLYMERS FOR ANTIFOULING SURFACES UNIV NORTHWESTERN (US) 2015-01-07 EP disclosed
EP-2812347-A1 AUTOPHAGY-INDUCING PEPTIDE Board Of Regents, The University Of Texas System (US) 2014-12-17 EP disclosed
WO-2014149440-A1 AUTOPHAGY-INDUCING PEPTIDE ANALOGS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-09-25 WO disclosed
WO-2013158600-A1 MULTIVALENT PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING SAME NEW YORK UNIVERSITY (US) 2013-10-24 WO disclosed
WO-2013119377-A1 AUTOPHAGY-INDUCING PEPTIDE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-08-15 WO disclosed
US-20120141997-A1 Compositions And Methods For Free-Solution Conjugate Nucleic Acid Analysis NORTHWESTERN UNIVERSITY (US) 2012-06-07 US disclosed
US-8114599-B2 Using multiplexed single-base extension assays comprising monodisperse uncharged polyamides conjugated to preferential nucleotide sequences for genotyping samples NORTHWESTERN UNIVERSITY (US) 2012-02-14 US disclosed
EP-2309850-A2 SURFACE-IMMOBILIZED ANTIMICROBIAL PEPTOIDS Northwestern University (US) 2011-04-20 EP disclosed
WO-2010014940-A2 SURFACE-IMMOBILIZED ANTIMICROBIAL PEPTOIDS NORTHWESTERN UNIVERSITY (US) 2010-02-04 WO disclosed
US-20100028719-A1 Surface-Immobilized Antimicrobial Peptoids NORTHWESTERN UNIVERSITY 2010-02-04 US disclosed
US-20090286435-A1 Method for Producing, and a Substrate with, a Surface with Specific Characteristics SURFACE INNOVATIONS LIMITED (GB) 2009-11-19 US disclosed
US-7618937-B2 Peptidomimetic polymers for antifouling surfaces NORTHWESTERN UNIVERSITY (US) 2009-11-17 US disclosed
US-20080241950-A1 Nucleic Acid Sequencing In Free Solution Using Protein Polymer Drag-Tags NORTHWESTERN UNIVERSITY (US) 2008-10-02 US disclosed
US-20080227211-A1 COMPOSITIONS AND METHODS FOR FREE-SOLUTION CONJUGATE NUCLEIC ACID ANALYSIS NORTHWESTERN UNIVERSITY (US) 2008-09-18 US disclosed
US-7371533-B2 Methods for separation of polymeric compounds UNIVERSITY OF OTTAWA (CA) 2008-05-13 US disclosed
EP-1868739-A2 METHOD FOR PRODUCING, AND A SUBSTRATE WITH, A SURFACE WITH SPECIFIC CHARACTERISTICS UNIVERSITY OF DURHAM (GB) 2007-12-26 EP disclosed
US-20070215472-A1 Electroosmotic flow for end labelled free solution electrophoresis UNIVERSITY OF OTTAWA (CA) 2007-09-20 US disclosed
EP-1814976-A2 PEPTIDOMIMETIC POLYMERS FOR ANTIFOULING SURFACES Northwestern University (US) 2007-08-08 EP disclosed
US-20060241281-A1 Peptidomimetic polymers for antifouling surfaces NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-10-26 US disclosed
WO-2006109055-A2 METHOD FOR COATING A SUBSTRATE TO GIVE PROTEIN RESISTANCE AND COATED SUBSTRATE UNIVERSITY OF DURHAM (GB) 2006-10-19 WO disclosed
US-20060177840-A1 Methods for separation of polymeric compounds DOE-DEITR 2006-08-10 US disclosed
WO-2006055531-A2 PEPTIDOMIMETIC POLYMERS FOR ANTIFOULING SURFACES NORTHWESTERN UNIVERSITY (US) 2006-05-26 WO disclosed
WO-2006055531-A2 PEPTIDOMIMETIC POLYMERS FOR ANTIFOULING SURFACES NORTHWESTERN UNIVERSITY (US) 2006-05-26 WO disclosed