SCHEMBL5992003

SCHEMBL5992003

CS(=O)(=O)c1ccc2oc3cc(Cl)ccc3c2c1Br

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AHR P35869 5/20 0.44
CCR2 P41597 8/20 0.42
MCL1 Q07820 1/20 0.38
TTR P02766 2/20 0.38
AKR1B1 P15121 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CDC25A P30304 1/20 0.35
CDC25C P30307 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5993039 0.81 AHR (0.53) AHRCCR2MCL1TTRAKR1B1
SCHEMBL20208693 0.72 AHR (0.63) AHRMCL1TTRCA1CA2
SCHEMBL29706029 0.72 AHR (0.63) AHRMCL1TTRCA1CA2
SCHEMBL5992006 0.71 AHR (0.49) AHRCCR2MCL1TTRCA1
SCHEMBL26502486 0.68 AHR (0.63) AHRMCL1TTRCA1CA2
SCHEMBL22737968 0.68 AHR (0.78) AHRMCL1TTRCA1CA2
SCHEMBL20208783 0.68 AHR (0.60) AHRMCL1TTRCA1CA2
SCHEMBL29706073 0.68 AHR (0.60) AHRMCL1TTRCA1CA2
SCHEMBL21191893 0.67 AHR (0.59) AHRMCL1TTRCA12CA1
SCHEMBL30409875 0.66 AHR (0.81) AHRTTRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735300-A1 THIO-SUBSTITUTED TRICYCLIC AND BICYCLIC AROMATIC METHANESULFINYL DERIVATIVES CEPHALON FRANCE (FR) 2006-12-27 EP disclosed
WO-2005100345-A1 THIO-SUBSTITUTED TRICYCLIC AND BICYCLIC AROMATIC METHANESULFINYL DERIVATIVES CEPHALON FRANCE (FR) 2005-10-27 WO disclosed