SCHEMBL5992695

SCHEMBL5992695

CCCS(=O)(=O)NC[C@H](C)c1ccc(-c2ccc([C@@H](C)CNS(=O)(=O)CCC)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 19/20 0.71
GRIA1 P42261 1/20 0.51
GRIA2 P42262 1/20 0.51
GRIA3 P42263 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565123 0.95 GRIA4 (0.68) GRIA4GRIA1GRIA2GRIA3
SCHEMBL27629410 0.90 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL27649580 0.90 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL27649556 0.90 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL7031129 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL6554706 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL6936169 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL6555617 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL6847064 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3
SCHEMBL6554686 0.87 GRIA4 (0.60) GRIA4GRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984756-B2 Process for preparing biphenyl compounds ELI LILLY AND COMPANY (US) 2006-01-10 US disclosed
US-20040235957-A1 Use of sulfonamide derivatives as pharmaceuticals compounds BLEAKMAN DAVID (US) 2004-11-25 US disclosed
US-20030225163-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225163-A1 Sulfonamide derivatives GRIN1, SLC1A2, GRIN2A GRIA4 17/4885GRIA1 8/4885GRIA2 10/4885
US-20040235957-A1 Use of sulfonamide derivatives as pharmaceuticals compounds GABRE, SCN2A, SCN1A GRIA4 212/4885GRIA1 324/4885GRIA2 176/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.