SCHEMBL5995877

SCHEMBL5995877

Nc1cccc2[nH]nc(C(=O)NC3CN4CCC3CC4)c12

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 8/20 0.71
HTR3A P46098 4/20 0.71
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1967617 1.00 CHRNA7 (0.71) CHRNA7HTR3AHTR3EHTR3BALOX15
SCHEMBL4602656 0.88 CHRNA7 (0.72) CHRNA7HTR3AHTR3EHTR3BALOX15
SCHEMBL492614 0.88 CHRNA7 (0.72) CHRNA7HTR3AHTR3EHTR3BALOX15
SCHEMBL492356 0.84 CHRNA7 (0.67) CHRNA7HTR3AHTR3EHTR3BHTR3D
SCHEMBL4605759 0.84 CHRNA7 (0.67) CHRNA7HTR3AHTR3EHTR3BHTR3D
SCHEMBL1964462 0.83 CHRNA7 (0.69) CHRNA7HTR3AHTR3EHTR3BALOX15
SCHEMBL5997237 0.83 CHRNA7 (0.69) CHRNA7HTR3AHTR3EHTR3BALOX15
Facinicline SCHEMBL260422 0.83 CHRNA7 (1.00) CHRNA7HTR3A
Facinicline SCHEMBL29749748 0.83 CHRNA7 (1.00) CHRNA7HTR3A
Facinicline SCHEMBL29365997 0.83 CHRNA7 (1.00) CHRNA7HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735306-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2006-12-27 EP disclosed
WO-2005092890-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed