Cpg-52852

Cpg-52852

SCHEMBL5999996

CCOCc1nc2c(N)nc3ccccc3c2n1CC(C)(C)NS(C)(=O)=O.CCc1nc2c(N)nc3ccccc3c2n1CCCCNS(C)(=O)=O

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TLR7

The experimentally established mechanism targets of Cpg-52852. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TLR7 known ✓ Q9NYK1 19/20 0.73
TLR8 Q9NR97 12/20 0.59
NUDT1 P36639 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2744632 0.90 TLR7 (0.81) TLR7TLR8NUDT1
SCHEMBL29421427 0.89 TLR7 (0.73) TLR7TLR8NUDT1
SCHEMBL29421426 0.89 TLR7 (0.73) TLR7TLR8NUDT1
SCHEMBL1616712 0.89 TLR7 (0.73) TLR7TLR8NUDT1
Water SCHEMBL4531043 0.88 TLR7 (0.72) TLR7TLR8NUDT1
SCHEMBL3968461 0.87 TLR7 (0.76) TLR7TLR8NUDT1
Cpg-52852 SCHEMBL483385 0.85 TLR7 (1.00) TLR7TLR8
Cpg-52852 SCHEMBL29371102 0.85 TLR7 (1.00) TLR7TLR8
SCHEMBL6000001 0.85 TLR7 (0.63) TLR7TLR8NUDT1
SCHEMBL728616 0.84 TLR7 (0.69) TLR7TLR8NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8961477-B2 Delivery of immune response modifier compounds 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-02-24 US disclosed
US-20060195067-A1 Delivery of immune response modifier compounds 3M INNOVATIVE PROPERTIES COMPANY 2006-08-31 US disclosed