SCHEMBL6003097

SCHEMBL6003097

O=C(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCN(CCN2[C@H](CO)CCC[C@@H]2CO)C[C@H]1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.48
RHOC P08134 1/20 0.44
RHOA P61586 1/20 0.44
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003101 1.00 TACR1 (0.48) TACR1RHOCRHOAKCNH2HRH3
Hydrochloric Acid SCHEMBL5368530 0.99 TACR1 (0.48) TACR1RHOCRHOAKCNH2HRH3
Hydrochloric Acid SCHEMBL5368523 0.99 TACR1 (0.48) TACR1RHOCRHOAKCNH2HRH3
Hydrochloric Acid SCHEMBL5369016 0.89 TACR1 (0.47) TACR1RHOCRHOA
Hydrochloric Acid SCHEMBL6003074 0.89 TACR1 (0.45) TACR1RHOCRHOA
Hydrochloric Acid SCHEMBL5526636 0.89 TACR1 (0.45) TACR1RHOCRHOA
Hydrochloric Acid SCHEMBL5366774 0.89 TACR1 (0.45) TACR1RHOCRHOA
Hydrochloric Acid SCHEMBL5366243 0.87 TACR1 (0.43) TACR1RHOCRHOA
Hydrochloric Acid SCHEMBL5366235 0.87 TACR1 (0.43) TACR1RHOCRHOA
SCHEMBL5360994 0.86 TACR1 (0.53) TACR1RHOCRHOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140924-B1 PIPERAZINE DERIVATIVES ASTELLAS PHARMA INC (JP) 2006-03-22 EP disclosed