SCHEMBL6003401

SCHEMBL6003401

O=C(c1ccc(OCCC2CCCCN2)cc1)c1c(-c2c(F)cc(F)cc2F)ccc2cc(O)ccc12

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.44
ESR1 P03372 17/20 0.41
ESR2 Q92731 16/20 0.41
SSTR2 P30874 1/20 0.36
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003304 0.99 CHEK2 (0.43) CHEK2ESR1ESR2
SCHEMBL6005869 0.93 CHEK2 (0.44) CHEK2ESR1ESR2SSTR2
SCHEMBL6004671 0.92 CHEK2 (0.43) CHEK2ESR1ESR2
SCHEMBL6004626 0.92 CHEK2 (0.44) CHEK2ESR1ESR2LTA4H
SCHEMBL6005392 0.91 ESR1 (0.42) CHEK2ESR1ESR2
SCHEMBL6003358 0.91 CHEK2 (0.43) CHEK2ESR1ESR2SSTR2LTA4H
Hydrochloric Acid SCHEMBL6003391 0.91 CHEK2 (0.43) CHEK2ESR1ESR2LTA4H
SCHEMBL6005357 0.91 CHEK2 (0.43) CHEK2ESR1ESR2LTA4H
SCHEMBL6003280 0.90 CHEK2 (0.43) CHEK2ESR1ESR2
SCHEMBL6004611 0.90 CHEK2 (0.43) CHEK2ESR1ESR2SSTR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709021-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2006-10-11 EP disclosed
WO-2005073204-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2005-08-11 WO disclosed