SCHEMBL6005134

SCHEMBL6005134

Oc1ccc2c(C(O)c3ccc(OCCC4CCCCCN4)cc3)c(-c3cc(F)ccc3F)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.42
ESR2 Q92731 14/20 0.42
LTA4H P09960 1/20 0.37
CHEK2 O96017 1/20 0.36
SSTR2 P30874 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004700 0.94 ESR1 (0.40) ESR1ESR2LTA4HCHEK2SSTR2
SCHEMBL6003243 0.91 ESR1 (0.41) ESR1ESR2LTA4HCHEK2SSTR2
SCHEMBL6005517 0.90 ESR1 (0.41) ESR1ESR2LTA4HCHEK2SSTR2
SCHEMBL6005667 0.89 ESR1 (0.40) ESR1ESR2LTA4HCHEK2SSTR2
Hydrochloric Acid SCHEMBL6005550 0.84 ESR1 (0.54) ESR1ESR2LTA4H
SCHEMBL6003362 0.83 CHEK2 (0.43) ESR1ESR2CHEK2
SCHEMBL1359346 0.83 ESR1 (0.62) ESR1ESR2
Hydrochloric Acid SCHEMBL6004757 0.82 ESR1 (0.49) ESR1ESR2LTA4HCHEK2SSTR2
SCHEMBL6003282 0.82 CHEK2 (0.43) ESR1ESR2LTA4HCHEK2
Hydrochloric Acid SCHEMBL6005706 0.79 ESR1 (0.54) ESR1ESR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709021-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2006-10-11 EP disclosed
WO-2005073204-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2005-08-11 WO disclosed