SCHEMBL6013246

SCHEMBL6013246

O=C(O)C1CNc2ncccc2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 12/20 0.43
KDM4E B2RXH2 1/20 0.38
CYP2C19 P33261 1/20 0.38
FAAH O00519 2/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRR1 P24046 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
GABRE P78334 1/20 0.37
GABRA6 Q16445 1/20 0.37
GABRG1 Q8N1C3 1/20 0.37
GABRG3 Q99928 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30585791 1.00 IDH1 (0.43) IDH1KDM4ECYP2C19FAAHGABRP
SCHEMBL28149742 0.86 IDH1 (0.42) IDH1KDM4EFAAH
SCHEMBL9805863 0.82 IDH1 (0.40) IDH1FAAH
SCHEMBL29550106 0.75 MAPT (0.56) IDH1KDM4EGAAMAPT
SCHEMBL2608547 0.75 MAPT (0.56) IDH1KDM4EGAAMAPT
SCHEMBL16464958 0.75 MAPT (0.56) IDH1KDM4EGAAMAPT
SCHEMBL16464959 0.75 MAPT (0.56) IDH1KDM4EGAAMAPT
SCHEMBL30288898 0.75 GAA (0.54) IDH1FAAHGABRPGABRDGABRA1
SCHEMBL924219 0.75 GAA (0.54) IDH1FAAHGABRPGABRDGABRA1
SCHEMBL29463686 0.75 GAA (0.54) IDH1FAAHGABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1684754-A1 HMG-COA REDUCTASE INHIBITORS AND METHOD Bristol-Myers Squibb Company (US) 2006-08-02 EP disclosed
WO-2005051386-A1 HMG-COA REDUCTASE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2005-06-09 WO disclosed