SCHEMBL6013738

SCHEMBL6013738

NCCn1c(-c2sccc2Cl)c(Cl)c2nc[nH]c(=O)c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.34
AURKA O14965 2/20 0.34
DAPK3 O43293 2/20 0.34
PRKD3 O94806 2/20 0.34
MAP4K4 O95819 2/20 0.34
RET P07949 2/20 0.34
IGF1R P08069 2/20 0.34
PIM1 P11309 2/20 0.34
CLK2 P49760 2/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
PRKX P51817 2/20 0.34
BTK Q06187 2/20 0.34
TYRO3 Q06418 2/20 0.34
DYRK1A Q13627 2/20 0.34
NTRK3 Q16288 2/20 0.34
TAOK1 Q7L7X3 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
ALK Q9UM73 2/20 0.34
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4335293 0.99 PARP1 (0.33) PARP1AURKADAPK3PRKD3MAP4K4
SCHEMBL6013734 0.89 AURKA (0.33) PARP1AURKADAPK3PRKD3MAP4K4
SCHEMBL13783369 0.89 PARP1 (0.35) PARP1AURKADAPK3PRKD3MAP4K4
Hydrochloric Acid SCHEMBL4344197 0.88 AURKA (0.32) PARP1AURKADAPK3PRKD3MAP4K4
Hydrochloric Acid SCHEMBL4334320 0.88 AURKA (0.34) PARP1AURKADAPK3PRKD3MAP4K4
SCHEMBL13843440 0.86 HTT (0.38) PARP1AURKADAPK3PRKD3MAP4K4
Hydrochloric Acid SCHEMBL3940563 0.85 HTT (0.38) PARP1AURKADAPK3PRKD3MAP4K4
SCHEMBL4330618 0.81 HPGD (0.38) PARP1AURKADAPK3PRKD3MAP4K4
Trifluoroacetic Acid SCHEMBL5983758 0.81 HRH4 (0.31) BRD4
Hydrochloric Acid SCHEMBL4323840 0.81 HPGD (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1661897-B1 PYRROLOPYRIMIDINONE DERIVATIVE TEIJIN PHARMA LTD (JP) 2013-12-04 EP disclosed
US-7557113-B2 Substituted pyrrolo[3,2-d]pyrimidine derivatives TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
US-7557113-B2 Substituted pyrrolo[3,2-d]pyrimidine derivatives TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
EP-1661897-A1 PYRROLOPYRIMIDINONE DERIVATIVE Teijin Pharma Limited (JP) 2006-05-31 EP disclosed