SCHEMBL6014057

SCHEMBL6014057

CN1CCC(Cc2ccc([C]=O)cc2C(F)(F)F)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 1/20 0.46
NR1H2 P55055 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
SSTR4 P31391 1/20 0.39
HTR2A P28223 3/20 0.36
ACHE P22303 3/20 0.35
BCHE P06276 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR2B P41595 1/20 0.34
MAPK14 Q16539 1/20 0.34
P2RX7 Q99572 1/20 0.34
CHEK1 O14757 1/20 0.34
SRC P12931 1/20 0.33
TAF1 P21675 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12426560 0.81 DDR1 (0.46) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL272847 0.80 NR1H2 (0.63) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL6014060 0.80 DDR1 (0.46) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL19178335 0.79 NR1H2 (0.65) NR1H2SRC
SCHEMBL3557511 0.79 DDR1 (0.56) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL272846 0.78 DDR1 (0.55) DDR1NR1H2NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL3555518 0.77 DDR1 (0.57) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL19072901 0.75 DDR1 (0.51) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL19073475 0.75 DDR1 (0.53) DDR1NR1H2NOS3NOS1NOS2
SCHEMBL29958951 0.75 DDR1 (0.49) DDR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299358-A1 AMIDE DERIVATIVE AND MEDICINE Nippon Shinyaku Co., Ltd. (JP) 2018-03-28 EP disclosed
EP-1702917-B1 AMIDE DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2017-08-02 EP disclosed
EP-1702917-A1 AMIDE DERIVATIVE AND MEDICINE Nippon Shinyaku Co., Ltd. (JP) 2006-09-20 EP disclosed