SCHEMBL6014681

SCHEMBL6014681

Nc1nc(-c2cccc(OCc3ccccc3)c2)cn2c1cnc2[C@H]1CC[C@H](CO)CC1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 18/20 0.53
TNK2 Q07912 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6014608 0.90 IGF1R (0.47) IGF1RTNK2
SCHEMBL5415358 0.89 IGF1R (0.50) IGF1RTNK2
SCHEMBL6014743 0.89 IGF1R (0.57) IGF1RTNK2
SCHEMBL6014690 0.86 IGF1R (0.49) IGF1RTNK2
SCHEMBL5114672 0.83 IGF1R (0.57) IGF1RTNK2
SCHEMBL5400865 0.83 IGF1R (0.43) IGF1RTNK2
SCHEMBL5394889 0.83 IGF1R (0.48) IGF1RTNK2
SCHEMBL1566947 0.77 TNK2 (0.38) IGF1RTNK2
SCHEMBL401018 0.77 TNK2 (0.38) IGF1RTNK2
SCHEMBL5390468 0.77 IGF1R (0.49) IGF1RTNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675860-A2 IMIDAZO[1,5-A]PYRAZINE TYROSINE KINASE INHIBITORS OSI Pharmaceuticals, Inc. (US) 2006-07-05 EP disclosed
WO-2005037836-A2 IMIDAZO ‘1, 5 - A ! PYRAZINE TYROSINE KINASE INHIBITORS OSI PHARMACEUTICALS, INC. (US) 2005-04-28 WO disclosed