SCHEMBL6016706

SCHEMBL6016706

CC[C@H](CO)Nc1nc(NCc2ccc(O)cc2)c2ncn(C(C)C)c2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 13/20 1.00
CCNB1 P14635 8/20 1.00
CCNB2 O95067 5/20 1.00
CCNB3 Q8WWL7 5/20 1.00
CDK2 P24941 9/20 0.84
CCNE1 P24864 8/20 0.84
CCNK O75909 8/20 0.84
CDK12 Q9NYV4 8/20 0.84
CDK5 Q00535 8/20 0.84
CDK7 P50613 6/20 0.84
CDK9 P50750 6/20 0.84
CDK4 P11802 4/20 0.84
CCND1 P24385 4/20 0.84
CCNH P51946 4/20 0.84
DYRK1A Q13627 3/20 0.84
MAPK1 P28482 3/20 0.84
CCNA2 P20248 3/20 0.84
CCNT1 O60563 3/20 0.84
CDK5R1 Q15078 3/20 0.84
CSNK1D P48730 2/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(Rs)-Roscovitine SCHEMBL172593 0.91 CDK1 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
Seliciclib SCHEMBL94728 0.91 CDK1 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
(Rs)-Roscovitine SCHEMBL15163619 0.91 CDK1 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
(S)-Roscovitine SCHEMBL2907488 0.91 CDK1 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
(S)-Roscovitine SCHEMBL29415376 0.91 CDK1 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL4501614 0.90 CDK2 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3877470 0.90 CDK2 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL2907920 0.90 CDK1 (0.81) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL17628573 0.90 CDK2 (1.00) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL1443401 0.90 CDK1 (0.85) CDK1CCNB1CCNB2CCNB3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244668-B1 PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF UNIVERSITAIRE INSTELLING ANTWE (BE) 2006-04-05 EP disclosed