SCHEMBL6018441

SCHEMBL6018441

CC(C)(C)OC(=O)N(Cc1ccc(C(=O)[C@H](CCCNCc2ncc[nH]2)C(=O)O)cc1)Cc1ccccn1.NCc1cccc2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.36
HDAC1 Q13547 3/20 0.35
HDAC3 O15379 2/20 0.35
HDAC2 Q92769 2/20 0.35
NCOR2 Q9Y618 2/20 0.35
FNTA P49354 2/20 0.35
FNTB P49356 2/20 0.35
BACE1 P56817 1/20 0.33
NAMPT P43490 1/20 0.33
MCL1 Q07820 1/20 0.33
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
F7 P08709 1/20 0.32
PGGT1B P53609 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
FOLH1 Q04609 1/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
KMT2A Q03164 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6018348 0.92 HDAC1 (0.35) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6018508 0.90 HDAC1 (0.35) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6018171 0.89 HDAC1 (0.35) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6019642 0.88 HDAC1 (0.34) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6018701 0.88 HDAC1 (0.34) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6018156 0.86 GCGR (0.34) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6690903 0.84 CXCR4 (0.41) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6019678 0.80 CXCR4 (0.46) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6689236 0.80 CXCR4 (0.40) CXCR4HDAC1HDAC3HDAC2NCOR2
SCHEMBL6018252 0.78 HDAC1 (0.44) HDAC1HDAC3HDAC2NCOR2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7098215-B2 Nitrogenous compounds and antiviral drugs containing the same KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2006-08-29 US disclosed
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same KUREHA CORPORATION (JP) 2004-05-13 US disclosed
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed
EP-1273571-A1 NITROGENOUS COMPOUNDS AND ANTIVIRAL DRUGS CONTAINING THE SAME Kureha Chemical Industry Co., Ltd. (JP) 2003-01-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same NSUN2, ZC3HAV1L, PNP CXCR4 2185/4885HDAC1 651/4885HDAC3 2307/4885
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 CXCR4 1/4885HDAC1 1092/4885HDAC3 1135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.