SCHEMBL6024708

SCHEMBL6024708

Cc1cc(C(=O)N2Cc3cnn(C)c3Nc3ccccc32)ccc1C#N.[O-][S+](Cl)Cl

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 19/20 0.62
OXTR P30559 13/20 0.62
AVPR2 P30518 7/20 0.62
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM3 P20309 1/20 0.47
DRD3 P35462 1/20 0.47
OPRK1 P41145 1/20 0.47
TSPO P30536 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4831821 0.95 AVPR1A (0.68) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2130334 0.85 AVPR1A (0.58) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL26185549 0.84 AVPR1A (0.75) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL30046134 0.84 AVPR1A (0.75) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18917272 0.81 AVPR1A (0.70) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL30045591 0.80 AVPR1A (0.69) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL26185571 0.80 AVPR1A (0.69) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL26564046 0.80 AVPR1A (0.69) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944536 0.79 AVPR1A (0.80) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL20277787 0.79 AVPR1A (0.66) AVPR1AOXTRAVPR2TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660501-A2 PIPERAZINES AS OXYTOCIN AGONISTS FERRING B.V. (NL) 2006-05-31 EP disclosed
WO-2005023812-A2 PIPERAZINES AS OXYTOCIN AGONISTS FERRING B.V. (NL) 2005-03-17 WO disclosed