SCHEMBL6027745

SCHEMBL6027745

Cc1cnc(C(=O)n2cc(Cl)c(C)n2)c(C)c1Br

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
ELANE P08246 3/20 0.32
ALDH1A1 P00352 1/20 0.32
MCL1 Q07820 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
PLAU P00749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395178 0.69 HSP90AA1 (0.44) HSP90AA1HSP90AB1
SCHEMBL11556929 0.67 KMT2A (0.32) MEN1KMT2ALMNAELANE
Hydrochloric Acid SCHEMBL11558888 0.66 MEN1 (0.33) MEN1KMT2ALMNAELANEALDH1A1
SCHEMBL3395737 0.64 HSP90AA1 (0.46) HSP90AA1HSP90AB1
SCHEMBL3395599 0.64 HSP90AA1 (0.47) HSP90AA1HSP90AB1
SCHEMBL28330033 0.63 HCAR2 (0.39) MEN1KMT2AALDH1A1MCL1
SCHEMBL14438199 0.62 CCR1 (0.37) LMNAHSP90AA1HSP90AB1
SCHEMBL28658089 0.61 HSP90AA1 (0.39) ALDH1A1HSP90AA1HSP90AB1
SCHEMBL1395393 0.60 HSP90AB1 (0.46) HSP90AA1HSP90AB1
Zinc Ion SCHEMBL10992139 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670802-A2 NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS Conforma Therapeutic Corporation (US) 2006-06-21 EP disclosed
WO-2005028434-A2 NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS CONFORMA THERAPEUTICS CORPORATION (US) 2005-03-31 WO disclosed