SCHEMBL6028154

SCHEMBL6028154

Cc1nc2cc(OCC(O)CN3CCN(CCOc4ccc(Br)c(Cl)c4)CC3)ccc2s1

nearest known ligand 0.61

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4332718 1.00 CYP3A4 (0.56) CYP3A4
SCHEMBL4334659 0.90 CYP3A4 (0.56) CYP3A4
SCHEMBL4334506 0.89 CYP3A4 (0.59) CYP3A4
SCHEMBL6028488 0.89 CYP3A4 (0.59) CYP3A4
SCHEMBL4323875 0.89 CYP3A4 (0.58) CYP3A4
SCHEMBL6027484 0.87 CYP3A4 (0.63) CYP3A4
SCHEMBL4333287 0.87 CYP3A4 (0.64) CYP3A4
SCHEMBL4327396 0.87 CYP3A4 (0.60) CYP3A4
SCHEMBL4329406 0.86 CYP3A4 (0.59) CYP3A4
SCHEMBL5405904 0.86 CYP3A4 (0.43) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723129-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2006-11-22 EP disclosed
WO-2005061470-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2005-07-07 WO disclosed