SCHEMBL6028301

SCHEMBL6028301

CCCCN1CCC(c2cc3cccc(C(N)=O)c3[nH]2)CC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.53
PARP2 Q9UGN5 1/20 0.53
AURKA O14965 2/20 0.46
AURKB Q96GD4 2/20 0.46
HTR1A P08908 2/20 0.43
DRD1 P21728 2/20 0.43
DRD4 P21917 2/20 0.43
DRD5 P21918 2/20 0.43
DRD3 P35462 2/20 0.43
DRD2 P14416 1/20 0.43
BTK Q06187 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29709485 0.94 PARP1 (0.60) PARP1PARP2DRD3DRD2
SCHEMBL6028914 0.94 PARP1 (0.60) PARP1PARP2DRD3DRD2
SCHEMBL6028177 0.85 PARP1 (0.56) PARP1PARP2
SCHEMBL5076303 0.83 PARP1 (0.55) PARP1PARP2AURKAAURKBHTR1A
SCHEMBL6028534 0.82 PARP1 (0.48) PARP1DRD4DRD3DRD2
SCHEMBL6029106 0.80 PARP1 (0.58) PARP1PARP2
Hydrochloric Acid SCHEMBL18614327 0.80 PARP1 (0.62) PARP1PARP2AURKAAURKB
SCHEMBL8818276 0.78 HRH3 (0.45) HTR1ADRD1DRD4DRD5DRD3
SCHEMBL5621656 0.78 PARP1 (0.62) PARP1PARP2AURKAAURKB
SCHEMBL6028492 0.78 PDPK1 (0.44) PARP1AURKABTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7087637-B2 Substituted indoles which are PARP inhibitors BASF AG (DE) 2006-08-08 US disclosed
US-20040067949-A1 Substituted indoles which are parp inhibitors ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2004-04-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040067949-A1 Substituted indoles which are parp inhibitors PARP1, PARP2, PARP12 PARP1 1/4885PARP2 2/4885AURKA 309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.