SCHEMBL6028339

SCHEMBL6028339

Cc1nc(C#Cc2cccc(Cl)c2)c[nH]1.Cc1nc(C#Cc2cccc(Cl)c2)cn1-c1ccoc1

nearest known ligand 0.44

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 16/20 0.44
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023081 0.91 GRM5 (0.50) GRM5KCNH2
SCHEMBL980685 0.80 GRM5 (0.61) GRM5KCNH2
SCHEMBL979991 0.74 GRM5 (0.48) GRM5KCNH2
SCHEMBL980654 0.74 GRM5 (0.58) GRM5KCNH2
SCHEMBL1020277 0.72 GRM5 (0.50) GRM5KCNH2
SCHEMBL1023078 0.71 GRM5 (0.53) GRM5KCNH2
SCHEMBL1021161 0.71 GRM5 (0.53) GRM5KCNH2
SCHEMBL983538 0.71 GRM5 (0.50) GRM5KCNH2
SCHEMBL1020958 0.70 GRM5 (0.54) GRM5KCNH2
SCHEMBL1020977 0.70 GRM5 (0.63) GRM5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670784-A1 HETEROARYL-SUBSTITUTED IMDAZOLE DERIVATIVES AS GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-06-21 EP disclosed
WO-2004111040-A1 HETEROARYL-SUBSTITUTED IMDAZOLE DERIVATIVES AS GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-12-23 WO disclosed