SCHEMBL6030704

SCHEMBL6030704

CS(=O)(=O)c1nc2cc(OC[C@H](O)CN3CCN(C4CC(=O)N(c5nc6ccccc6o5)C4=O)CC3)ccc2s1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4334520 0.90 CYP3A4 (0.53) CYP3A4CYP1A2CYP2C9
SCHEMBL4328186 0.79 CYP3A4 (0.60) CYP3A4CYP1A2CYP2C9
SCHEMBL4334460 0.77 CYP3A4 (0.58) CYP3A4CYP1A2CYP2C9
SCHEMBL4327432 0.77 CYP3A4 (0.55) CYP3A4CYP1A2CYP2C9
SCHEMBL4342073 0.75 CYP3A4 (0.56) CYP3A4CYP1A2CYP2C9
SCHEMBL4326275 0.74 CYP3A4 (0.55) CYP3A4CYP1A2CYP2C9
SCHEMBL4329604 0.74 CYP3A4 (0.55) CYP3A4CYP1A2CYP2C9
SCHEMBL4334863 0.74 CYP3A4 (0.55) CYP3A4CYP1A2CYP2C9
SCHEMBL4329914 0.74 CYP3A4 (0.57) CYP3A4CYP1A2CYP2C9
SCHEMBL4333645 0.73 CYP3A4 (0.54) CYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723129-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2006-11-22 EP disclosed
WO-2005061470-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2005-07-07 WO disclosed