SCHEMBL6052097

SCHEMBL6052097

Cc1c(C(=O)Nc2ccc(N3CCC(N4CCOCC4)CC3)c(C#N)c2)cnn1-c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.49
RAB9A P51151 11/20 0.43
NPC1 O15118 9/20 0.43
PKM P14618 1/20 0.43
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43
MAPT P10636 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
POLB P06746 1/20 0.41
MITF O75030 1/20 0.41
G6PD P11413 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
MC4R P32245 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6052358 0.95 NR1H4 (0.46) NR1H4RAB9ANPC1PKMMAPK8
SCHEMBL6052244 0.92 MCHR1 (0.45) NR1H4RAB9ANPC1PKMMAPT
SCHEMBL31303184 0.92 MCHR1 (0.45) NR1H4RAB9ANPC1PKMMAPT
SCHEMBL6052562 0.92 NPC1 (0.52) NR1H4RAB9ANPC1PKMMAPT
Hydrochloric Acid SCHEMBL6052197 0.92 MCHR1 (0.44) NR1H4RAB9ANPC1PKMMAPT
SCHEMBL6052420 0.91 NR1H4 (0.45) NR1H4RAB9ANPC1PKMMAPT
Water SCHEMBL6052740 0.91 NR1H4 (0.45) NR1H4RAB9ANPC1PKMMAPT
SCHEMBL6052141 0.90 HTT (0.45) NR1H4RAB9ANPC1PKMMAPT
SCHEMBL6052617 0.90 RAF1 (0.47) NR1H4RAB9ANPC1
SCHEMBL6052406 0.89 NR1H4 (0.43) NR1H4RAB9ANPC1PKMMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7015218-B1 Amide compounds and medicinal use thereof MITSUBISHI PHARMA CORPORATION (JP) 2006-03-21 US claimed
EP-1176140-B1 AMIDE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI PHARMA CORP (JP) 2004-12-29 EP claimed
EP-1176140-A1 AMIDE COMPOUNDS AND MEDICINAL USE THEREOF Mitsubishi Pharma Corporation (JP) 2002-01-30 EP claimed
US-7015218-B1 Amide compounds and medicinal use thereof MITSUBISHI PHARMA CORPORATION (JP) 2006-03-21 US disclosed
EP-1176140-B1 AMIDE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI PHARMA CORP (JP) 2004-12-29 EP disclosed
EP-1176140-A1 AMIDE COMPOUNDS AND MEDICINAL USE THEREOF Mitsubishi Pharma Corporation (JP) 2002-01-30 EP disclosed