SCHEMBL6054773

SCHEMBL6054773

O=C1OC2(CCN(c3cnc(-c4ccccc4)cn3)CC2)c2ccc(F)cc21

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 2/20 0.54
NPY5R Q15761 14/20 0.51
DGAT1 O75907 2/20 0.45
KCNH2 Q12809 1/20 0.44
HSD11B1 P28845 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657710 0.87 NPY5R (0.64) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL4577444 0.83 AVPR1A (0.58) AVPR1ANPY5R
SCHEMBL6054873 0.82 AVPR1A (0.54) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL4164094 0.81 NPY5R (0.79) NPY5R
SCHEMBL4016619 0.79 NPY5R (0.48) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL4577327 0.79 NPY5R (0.57) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL4577476 0.79 NPY5R (0.55) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL6054824 0.78 NPY5R (0.66) AVPR1ANPY5RDGAT1HSD11B1
SCHEMBL4577315 0.73 NPY5R (0.81) NPY5R
SCHEMBL4158894 0.73 NPY5R (0.79) NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1635773-A2 COMBINATION THERAPY FOR THE TREATMENT OF HYPERTENSION Merck & Co., Inc. (a New Jersey corp.) (US) 2006-03-22 EP disclosed
WO-2004110368-A2 COMBINATION THERAPY FOR THE TREATMENT OF HYPERTENSION MERCK & CO., INC. (US) 2004-12-23 WO disclosed