SCHEMBL6058876

SCHEMBL6058876

CCOC(=O)C(Cc1ccnc(NC(=O)OC(C)(C)C)c1)C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 7/20 0.44
IGF1R P08069 1/20 0.42
PKM P14618 1/20 0.41
CYP17A1 P05093 1/20 0.40
MAPK14 Q16539 2/20 0.40
CCR2 P41597 2/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
PPARG P37231 1/20 0.39
MMP8 P22894 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6058886 0.95 NR3C2 (0.43) NR3C2IGF1RPKMCYP17A1MAPK14
SCHEMBL5079952 0.88 NR3C2 (0.48) NR3C2IGF1RCYP17A1CCR2PPARG
SCHEMBL190869 0.83 IGF1R (0.44) NR3C2IGF1RPKMCYP17A1MAPK14
SCHEMBL6058814 0.83 IGF1R (0.40) NR3C2IGF1RPKMCYP17A1MAPK14
SCHEMBL12596578 0.83 NR3C2 (0.47) NR3C2IGF1RCYP17A1CCR2
SCHEMBL12540360 0.83 NR3C2 (0.47) NR3C2IGF1RCYP17A1CCR2
SCHEMBL6058884 0.83 NR3C2 (0.42) NR3C2IGF1RCYP17A1MAPK14CCR2
SCHEMBL15354529 0.82 RIOK2 (0.50) NR3C2IGF1RPKMCYP17A1MAPK14
SCHEMBL6058751 0.82 NAMPT (0.44) PKMCYP17A1ALDH1A1GAAMKNK2
SCHEMBL21999119 0.81 NR3C2 (0.44) NR3C2IGF1RCYP17A1CCR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed