SCHEMBL6068433

SCHEMBL6068433

COc1cc(CNc2cc(N3CCOCC3)nc(Nc3nc(C)c(C(=O)O)s3)n2)cc(OC)c1OC

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 6/20 0.58
PIK3CB P42338 8/20 0.45
PIK3CA P42336 3/20 0.45
AURKA O14965 2/20 0.45
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
CRHBP P24387 1/20 0.40
HTT P42858 1/20 0.40
CRHR2 Q13324 1/20 0.40
PIK3CD O00329 1/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29831936 0.92 PDE5A (0.70) PDE5APIK3CBPIK3CAAURKAALDH1A1
SCHEMBL28578234 0.92 PDE5A (0.70) PDE5APIK3CBPIK3CAAURKAALDH1A1
SCHEMBL299684 0.91 PDE5A (0.70) PDE5APIK3CBPIK3CAAURKAKDM4E
SCHEMBL26647635 0.91 PDE5A (0.62) PDE5AAURKA
SCHEMBL289823 0.90 PDE5A (0.58) PDE5AAURKAALDH1A1KDM4ETSHR
SCHEMBL290275 0.89 PDE5A (0.57) PDE5AAURKAALDH1A1KDM4ETSHR
SCHEMBL291065 0.88 PDE5A (0.58) PDE5AAURKAALDH1A1KDM4ETSHR
SCHEMBL291323 0.88 PDE5A (0.56) PDE5AALDH1A1KDM4ETSHRMAPT
SCHEMBL27950935 0.84 PDE5A (0.49) PDE5APIK3CBPIK3CAALDH1A1KDM4E
SCHEMBL291180 0.84 PDE5A (0.54) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7087614-B2 Pyrimidine inhibitors of phosphodiesterase (PDE) 7 BRISTOL-MYERS SQUIBB CO. (US) 2006-08-08 US disclosed