SCHEMBL6068484

SCHEMBL6068484

Nc1nnc(C(=O)O)c2sc(-c3ccc(CN4CCOCC4)cc3)cc12

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 10/20 0.47
JAK1 P23458 9/20 0.47
TYK2 P29597 9/20 0.47
JAK3 P52333 8/20 0.47
KCNH2 Q12809 4/20 0.43
HRH3 Q9Y5N1 2/20 0.43
PIK3CD O00329 1/20 0.41
PARP1 P09874 2/20 0.40
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6407476 0.92 JAK2 (0.52) JAK2JAK1TYK2JAK3KCNH2
SCHEMBL5458391 0.79 JAK2 (0.75) JAK2JAK1TYK2JAK3PARP1
SCHEMBL6068379 0.77 JAK2 (0.52) JAK2JAK1TYK2JAK3NPC1
SCHEMBL3510941 0.72 CHEK1 (0.56) JAK2JAK1TYK2JAK3KCNH2
SCHEMBL1926925 0.72 IKBKB (0.56) JAK2HRH3PARP1RAB9A
SCHEMBL11907261 0.71 PARP1 (0.59) JAK2HRH3PARP1HTTSMN1; SMN2
SCHEMBL30508238 0.69 LRRK2 (0.57) JAK2HRH3
SCHEMBL6401995 0.68 JAK2 (0.51) JAK2JAK1TYK2JAK3
SCHEMBL27586651 0.68 HTT (0.46) HRH3NPC1HTTRAB9ASMN1; SMN2
SCHEMBL254490 0.68 HRH3 (0.72) HRH3NPC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7135470-B2 Thienopyridazines as IKK inhibitors ROCHE PALO ALTO LLC (US) 2006-11-14 US disclosed