SCHEMBL6072704

SCHEMBL6072704

Cc1ccc2c(C(CO)c3ccccn3)c(CCN(C)C)sc2c1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 18/20 0.58
CYP2D6 P10635 11/20 0.58
KCNH2 Q12809 10/20 0.58
CHRM1 P11229 5/20 0.58
CYP3A4 P08684 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072944 0.88 HRH1 (0.73) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL4843783 0.86 HRH1 (0.78) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL4846590 0.86 HRH1 (0.78) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL4846478 0.86 HRH1 (0.78) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072986 0.80 HRH1 (0.50) HRH1CYP2D6KCNH2CHRM1
SCHEMBL6072703 0.80 HRH1 (0.52) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072724 0.79 HRH1 (0.63) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL4849055 0.75 HRH1 (0.77) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072671 0.74 HRH1 (0.76) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072709 0.74 HRH1 (0.74) HRH1CYP2D6KCNH2CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO claimed
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO disclosed