SCHEMBL6072964

SCHEMBL6072964

Cc1ccc(CC(O)c2c(CCN(C)C)sc3ccccc23)cn1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 19/20 0.68
CYP2D6 P10635 12/20 0.56
KCNH2 Q12809 9/20 0.56
CHRM1 P11229 7/20 0.54
CYP3A4 P08684 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072803 0.83 HRH1 (0.63) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072714 0.81 HRH1 (0.64) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072942 0.81 HRH1 (0.64) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL4846545 0.81 HRH1 (1.00) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072967 0.81 HRH1 (0.75) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072789 0.81 HRH1 (0.67) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072718 0.81 HRH1 (0.65) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072666 0.80 HRH1 (0.66) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072707 0.79 HRH1 (0.65) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6072817 0.79 HRH1 (0.65) HRH1CYP2D6KCNH2CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO claimed
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO disclosed