SCHEMBL6089436

SCHEMBL6089436

OCc1cncn1Cc1ccc2ccccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.45
CYP11B2 P19099 3/20 0.45
CYSLTR1 Q9Y271 3/20 0.42
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
GPBAR1 Q8TDU6 2/20 0.39
FAAH O00519 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYSLTR2 Q9NS75 1/20 0.38
AKR1B1 P15121 1/20 0.38
QPCT Q16769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7459241 0.92 CYP11B1 (0.42) CYP11B1CYP11B2CYSLTR1HDAC3HDAC4
SCHEMBL6599637 0.75 CYP11B1 (0.56) CYP11B1CYP11B2
SCHEMBL3079356 0.73 CYP11B1 (0.71) CYP11B1CYP11B2
SCHEMBL6923450 0.72 CYP2C19 (0.53) CYP11B1CYP11B2
SCHEMBL243295 0.72 CYSLTR1 (0.57) CYSLTR1GPBAR1CYP1A2CYSLTR2
SCHEMBL28496074 0.70 CYSLTR1 (0.56) CYSLTR1GPBAR1CYP1A2CYSLTR2
Hydrochloric Acid SCHEMBL3129974 0.70 CYSLTR1 (0.56) CYSLTR1GPBAR1CYP1A2CYSLTR2
SCHEMBL17372091 0.70 CYP19A1 (0.44) CYSLTR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL6088426 0.70 CYSLTR1 (0.46) CYSLTR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL6928773 0.69 CYP11B1 (0.48) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed