SCHEMBL6090277

SCHEMBL6090277

CCN(CC)C(C)c1c(C)[nH]c(/C=C2/C(=O)NN=C2c2cccnc2)c1C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.47
CHEK1 O14757 2/20 0.47
ALK Q9UM73 4/20 0.39
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
ABL1 P00519 2/20 0.35
RET P07949 2/20 0.35
FLT3 P36888 2/20 0.35
PDGFRB P09619 3/20 0.31
FGFR1 P11362 2/20 0.30
PRKAA2 P54646 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PARP10 Q53GL7 1/20 0.30
PARP11 Q9NR21 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092863 0.89 KDR (0.44) KDRCHEK1ALDH1A1LMNAPDGFRB
SCHEMBL6089250 0.89 KDR (0.45) KDRCHEK1ALDH1A1LMNA
SCHEMBL6090063 0.84 KDR (0.45) KDRCHEK1ALKABL1RET
SCHEMBL6090365 0.84 KDR (0.66) KDRCHEK1
SCHEMBL6089341 0.84 KDR (0.46) KDRCHEK1ALKABL1RET
SCHEMBL6088780 0.81 KDR (0.49) KDRCHEK1ALKABL1RET
SCHEMBL6088845 0.81 KDR (0.59) KDRCHEK1ALKALDH1A1LMNA
SCHEMBL6088839 0.81 KDR (0.59) KDRCHEK1ALKALDH1A1LMNA
SCHEMBL6090868 0.80 KDR (0.41) KDRCHEK1PDGFRB
SCHEMBL6092350 0.80 KDR (0.41) KDRCHEK1ALKABL1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed