SCHEMBL6090381

SCHEMBL6090381

O=C1NN=C(c2cccnc2)/C1=C/c1ccc(C(F)(F)F)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.41
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
HSD17B4 P51659 1/20 0.40
KDR P35968 4/20 0.39
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
JAK3 P52333 4/20 0.35
JAK2 O60674 1/20 0.35
NPY5R Q15761 3/20 0.35
BTK Q06187 1/20 0.34
TYMP P19971 1/20 0.33
ERN1 O75460 1/20 0.33
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6090385 1.00 ALK (0.41) ALKHSD17B1HSD17B2HSD17B4KDR
SCHEMBL6090988 0.82 KDR (0.49) ALKKDRALDH1A1LMNAPDE3B
SCHEMBL6090995 0.82 KDR (0.49) ALKKDRALDH1A1LMNAPDE3B
SCHEMBL6089687 0.82 KDR (0.54) KDR
SCHEMBL6089692 0.82 KDR (0.54) KDR
SCHEMBL6102271 0.77 JAK3 (0.57) ALKKDRALDH1A1LMNAJAK3
SCHEMBL6102265 0.77 JAK3 (0.57) ALKKDRALDH1A1LMNAJAK3
SCHEMBL6091863 0.76 KDR (0.31) KDR
SCHEMBL6091867 0.76 KDR (0.31) KDR
SCHEMBL6093034 0.76 ALK (0.40) ALKKDRALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed