SCHEMBL6092111

SCHEMBL6092111

Cc1sc(C(=O)O)c2c1[C@H]1[C@@H](C2)C1(C)C.NCc1ccc(OCCCO)cc1Cl

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.71
S1PR3 Q99500 11/20 0.71
CACNA1G O43497 1/20 0.47
CACNA1H O95180 1/20 0.47
CACNA1I Q9P0X4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6093010 0.89 S1PR1 (0.70) S1PR1S1PR3
SCHEMBL1384889 0.88 S1PR1 (0.61) S1PR1S1PR3CACNA1GCACNA1HCACNA1I
SCHEMBL1381068 0.88 S1PR1 (0.61) S1PR1S1PR3CACNA1GCACNA1HCACNA1I
SCHEMBL2949720 0.86 S1PR1 (0.93) S1PR1S1PR3
SCHEMBL6111416 0.86 S1PR1 (0.68) S1PR1S1PR3
SCHEMBL2941999 0.85 S1PR1 (0.75) S1PR1S1PR3CACNA1GCACNA1HCACNA1I
SCHEMBL6090755 0.85 S1PR1 (0.76) S1PR1S1PR3
SCHEMBL5226138 0.84 S1PR1 (0.54) S1PR1S1PR3CACNA1GCACNA1HCACNA1I
SCHEMBL2948159 0.83 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL2943034 0.81 S1PR1 (0.80) S1PR1S1PR3CACNA1GCACNA1HCACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006010379-A1 NOVEL THIOPHENE DERIVATIVES AS IMMUNOSUPPRESSIVE AGENTS ACTELION PHARMACEUTICALS LTD. (CH) 2006-02-02 WO disclosed