SCHEMBL6095059

SCHEMBL6095059

Cc1nn(-c2ccc(CCO)cc2)c(C)c1-c1cc(F)cc(F)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 1/20 0.44
AR P10275 4/20 0.42
PTGS2 P35354 1/20 0.38
TP53 P04637 2/20 0.38
LMNA P02545 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
KMT2A Q03164 1/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6096797 0.88 CYP1A2 (0.72) CYP1A2CYP2D6ARPTGS2TP53
SCHEMBL6097347 0.87 CYP1A2 (0.63) CYP1A2CYP2D6ARLMNARAB9A
SCHEMBL6097885 0.87 CYP1A2 (0.56) CYP1A2CYP2D6ARTP53LMNA
SCHEMBL6097549 0.85 CYP1A2 (0.56) CYP1A2CYP2D6ARPTGS2TP53
SCHEMBL6097637 0.84 CYP1A2 (0.59) CYP1A2CYP2D6ARTP53LMNA
SCHEMBL6098575 0.83 CYP1A2 (0.53) CYP1A2TP53RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6096492 0.81 CYP1A2 (0.54) CYP1A2CYP2D6ARPTGS2TP53
SCHEMBL6098897 0.79 CYP1A2 (0.52) CYP1A2CYP2D6PTGS2LMNARAB9A
SCHEMBL6099027 0.78 SMN1; SMN2 (0.53) CYP1A2TP53LMNASMN1; SMN2
SCHEMBL6095421 0.77 CYP1A2 (0.50) CYP1A2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7001917-B2 Pyrazole compounds as anti-inflammatory and analgesic agents WARNER LAMBERT COMPANY LLC (US) 2006-02-21 US disclosed
US-20040019045-A1 2-(4-(4-(4-Fluorophenyl)-3,5-imethyl-1H-pyrazol-1-yl)phenyl) ethyl (4-methylphenyl)sulfonylcarbamate ammonium salt, e.g., as an antagonist for Prostoglandin E receptor; analgesics; antipyretics; antiinflammatory agents HIRANO MISATO (JP) 2004-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040019045-A1 2-(4-(4-(4-Fluorophenyl)-3,5-imethyl-1H-pyrazol-1-yl)phenyl) ethyl (4-methylphenyl)sulfonylcarbamate ammonium salt, e.g., as an antagonist for Prostoglandin E receptor; analgesics; antipyretics; antiinflammatory agents PTGER1, PTGS1, PTGIR CYP1A2 670/4885CYP2D6 801/4885AR 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.