SCHEMBL6099213

SCHEMBL6099213

Cc1[nH]c(C=C2C(=O)NN=C2c2nccnn2)c(C(C)C)c1CN1CCCC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.38
CHEK1 O14757 2/20 0.38
KMT2A Q03164 2/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6099201 1.00 KDR (0.38) KDRCHEK1KMT2AHSD17B10L3MBTL1
SCHEMBL6101257 0.92 KDR (0.38) KDRCHEK1KMT2AHSD17B10L3MBTL1
SCHEMBL6101240 0.92 KDR (0.38) KDRCHEK1KMT2AHSD17B10L3MBTL1
SCHEMBL6091384 0.91 KDR (0.38) KDRCHEK1
SCHEMBL6091392 0.91 KDR (0.38) KDRCHEK1
SCHEMBL6088165 0.89 KDR (0.37) KDRCHEK1
SCHEMBL6088180 0.89 KDR (0.37) KDRCHEK1
SCHEMBL6099584 0.85 KDR (0.38) KDRCHEK1KMT2AHSD17B10L3MBTL1
SCHEMBL6100513 0.85 KDR (0.55) KDRCHEK1KMT2AHSD17B10
SCHEMBL6099578 0.85 KDR (0.38) KDRCHEK1KMT2AHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP disclosed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed